SCHEMBL9705710

SCHEMBL9705710

Cc1cc(-c2nc(C)c(C)o2)cc(C)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
GAA P10253 2/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 1/20 0.34
ALOX5 P09917 4/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
PTPN1 P18031 1/20 0.34
KDM4E B2RXH2 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PTGS1 P23219 3/20 0.32
PTGS2 P35354 3/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2B6 P20813 1/20 0.32
TTR P02766 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9863203 0.80 SNCA (0.46) NPC1RAB9AMAPTESR1ESR2
SCHEMBL9862893 0.74 NPC1 (0.51) GAAKDM4ENPC1RAB9AMAPT
SCHEMBL3590075 0.73 HDAC6 (0.47) GAACYP1A2CYP2C9CYP2C19RAB9A
SCHEMBL11326576 0.70 NPC1 (0.55) GAAKDM4ENPC1RAB9APTGS2
SCHEMBL436384 0.69 GAA (0.57) GAAKDM4ENPC1RAB9AALDH1A1
SCHEMBL2706143 0.69 NPC1 (0.52) CYP1A2CYP2C9KDM4ENPC1RAB9A
SCHEMBL220910 0.68 CA1 (1.00) CA1CA2GAACYP1A2CYP2C9
SCHEMBL22804025 0.68 CA1 (1.00) CA1CA2GAACYP1A2CYP2C9
SCHEMBL13633790 0.68 TP53 (0.50) GAACYP1A2CYP2C19KDM4ENPC1
SCHEMBL14070535 0.68 CA1 (0.65) CA1CA2GAACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0207454-B1 ISOXAZOLE AND FURAN DERIVATIVES, THEIR PREPARATION AND USE AS ANTIVIRAL AGENTS STERLING WINTHROP INC. (US) 1992-09-09 EP disclosed
US-5002960-A Viricides for combating picornaviruses STERLING DRUG, INC. (US) 1991-03-26 US disclosed
US-4939267-A Viricides STERLING DRUG INC. (US) 1990-07-03 US disclosed
US-4843087-A OXAZOLINYL COMPOUNDS; RHINOVIRUSES AND PICORNAVIRUSES STERLING DRUG INC. (US) 1989-06-27 US disclosed
EP-0207454-A2 Isoxazole and furan derivatives, their preparation and use as antiviral agents STERLING WINTHROP INC. (US) 1987-01-07 EP disclosed