SCHEMBL9705741

SCHEMBL9705741

NC(=O)NC(=O)c1nc2cc(Cl)c(Cl)cc2[nH]c1=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 4/20 0.65
GRIN3B O60391 4/20 0.65
GRIA1 P42261 4/20 0.65
GRIA2 P42262 4/20 0.65
GRIA3 P42263 4/20 0.65
GRIA4 P48058 4/20 0.65
GRIN1 Q05586 4/20 0.65
GRIN2A Q12879 4/20 0.65
GRIN2B Q13224 4/20 0.65
GRIN2C Q14957 4/20 0.65
GRIN3A Q8TCU5 4/20 0.65
GRIK1 P39086 2/20 0.65
GRIK2 Q13002 2/20 0.65
GRIK3 Q13003 2/20 0.65
GRIK4 Q16099 2/20 0.65
GRIK5 Q16478 2/20 0.65
LMNA P02545 2/20 0.65
EGLN1 Q9GZT9 2/20 0.45
CACNA1G O43497 1/20 0.44
PRKAG1 P54619 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703410 0.86 GRIN2D (0.68) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9703949 0.84 GRIN2D (0.70) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9703926 0.84 GRIN2D (0.74) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9704899 0.83 GRIN2D (0.71) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9704115 0.82 GRIN2D (0.67) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9705036 0.82 GRIN2D (0.66) GRIN2DGRIN3BGRIA1GRIA2GRIA3
6,7-Dichloro-3-Hydroxy-2-Quinoxalinecarboxylic Acid SCHEMBL6697845 0.79 GRIN2D (1.00) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9704050 0.79 GRIN2D (0.62) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9704240 0.78 EGLN1 (0.70) GRIN2DGRIN3BGRIA1GRIA2GRIA3
SCHEMBL9704360 0.78 GRIN2D (1.00) GRIN2DGRIN3BGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011245-A1 2-ACYLAMIDO DERIVATIVES OF 3,4-DIHYDRO-3-OXO-QUINOXALINE HAVING PHARMACEUTICAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-07-09 WO disclosed