SCHEMBL9706487

SCHEMBL9706487

Cc1cccc(C)c1NCCn1ccnc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
QPCT Q16769 2/20 0.51
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
EGFR P00533 1/20 0.50
ALDH1A1 P00352 4/20 0.49
LMNA P02545 3/20 0.49
HPGD P15428 2/20 0.49
TSHR P16473 2/20 0.49
MAPK1 P28482 2/20 0.49
ALOX15 P16050 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
CASP1 P29466 1/20 0.48
CLK1 P49759 1/20 0.48
CASP7 P55210 1/20 0.48
HSD17B10 Q99714 1/20 0.48
SOD1 P00441 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706477 0.90 MEN1 (0.58) KMT2AMEN1QPCTEGFRALDH1A1
SCHEMBL20659412 0.84 CYP11B1 (0.53) KMT2AMEN1QPCTCYP11B1CYP11B2
SCHEMBL13164564 0.78 CYP1A2 (0.56) KMT2AMEN1QPCTCYP11B1CYP11B2
SCHEMBL9662466 0.76 KMT2A (0.49) KMT2AMEN1QPCTCYP11B1CYP11B2
SCHEMBL18457438 0.76 QPCT (0.56) QPCTCYP11B1CYP11B2POLBSOD1
SCHEMBL15933383 0.74 POLB (0.45) KMT2AMEN1QPCTLMNATSHR
SCHEMBL9706486 0.74 MEN1 (0.56) KMT2AMEN1ALDH1A1LMNAHPGD
Bromide SCHEMBL9706367 0.73 MEN1 (0.55) KMT2AMEN1ALDH1A1LMNAHPGD
SCHEMBL9323999 0.72 CYP11B1 (0.58) KMT2AMEN1CYP11B1CYP11B2ALDH1A1
SCHEMBL30674929 0.72 CYP11B1 (0.58) KMT2AMEN1CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0198325-B1 SUBSTITUTED ANILINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1992-07-15 EP disclosed
US-4891429-A CHEMICAL INTERMEDIATES HOFFMANN-LA ROCHE INC. (US) 1990-01-02 US disclosed
US-4696930-A CARDIOVASCULAR DISORDERS, ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1987-09-29 US disclosed
EP-0198325-A2 Substituted aniline derivatives F. HOFFMANN-LA ROCHE AG (CH) 1986-10-22 EP disclosed