SCHEMBL9706477

SCHEMBL9706477

Cc1cccc(C)c1NCCCCn1ccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
QPCT Q16769 2/20 0.57
LMNA P02545 3/20 0.55
ALDH1A1 P00352 3/20 0.55
TSHR P16473 3/20 0.55
MAPK1 P28482 2/20 0.55
HPGD P15428 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
ALOX15 P16050 1/20 0.55
EGFR P00533 1/20 0.55
KDM4E B2RXH2 1/20 0.54
POLB P06746 1/20 0.54
CASP1 P29466 1/20 0.54
CLK1 P49759 1/20 0.54
CASP7 P55210 1/20 0.54
HSD17B10 Q99714 1/20 0.54
SOD1 P00441 2/20 0.53
TBXAS1 P24557 1/20 0.50
PRKCI P41743 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706487 0.90 KMT2A (0.55) MEN1KMT2AQPCTLMNAALDH1A1
SCHEMBL20659412 0.80 CYP11B1 (0.53) MEN1KMT2AQPCTLMNAALDH1A1
SCHEMBL9706486 0.76 MEN1 (0.56) MEN1KMT2ALMNAALDH1A1TSHR
SCHEMBL5838710 0.76 MAPT (0.44) MEN1KMT2ALMNAALDH1A1TSHR
Bromide SCHEMBL9706367 0.75 MEN1 (0.55) MEN1KMT2ALMNAALDH1A1TSHR
SCHEMBL5551707 0.74 SOD1 (0.53) MEN1KMT2AQPCTALDH1A1SMN1; SMN2
SCHEMBL9849578 0.74 ALDH1A1 (0.61) MEN1KMT2AQPCTLMNAALDH1A1
SCHEMBL9849642 0.74 ALDH1A1 (0.61) MEN1KMT2AQPCTLMNAALDH1A1
SCHEMBL5839061 0.74 CHRM2 (0.44) MEN1KMT2AALDH1A1KDM4ECYP1A2
SCHEMBL10771358 0.73 TBXAS1 (0.67) QPCTHSD17B10TBXAS1PRKCICYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0198325-B1 SUBSTITUTED ANILINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1992-07-15 EP disclosed
US-4891429-A CHEMICAL INTERMEDIATES HOFFMANN-LA ROCHE INC. (US) 1990-01-02 US disclosed
US-4696930-A CARDIOVASCULAR DISORDERS, ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1987-09-29 US disclosed
EP-0198325-A2 Substituted aniline derivatives F. HOFFMANN-LA ROCHE AG (CH) 1986-10-22 EP disclosed