SCHEMBL9707366

SCHEMBL9707366

COC(=O)Cn1c(=O)n(CC(C)C)c(=O)c2c1nc(C1CCCCC1)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 8/20 0.39
AGTR2 P50052 4/20 0.39
PPARG P37231 3/20 0.38
KMT2A Q03164 2/20 0.36
ADORA3 P0DMS8 2/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
BLM P54132 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707929 0.97 AGTR1 (0.39) AGTR1AGTR2PPARGKMT2APOLB
SCHEMBL9707400 0.94 AGTR1 (0.42) AGTR1AGTR2PPARGKMT2APOLB
SCHEMBL9707886 0.93 PDE5A (0.43) AGTR1AGTR2PPARGKMT2A
SCHEMBL9708682 0.92 KMT2A (0.41) AGTR1AGTR2KMT2AADORA3POLB
SCHEMBL9707672 0.91 PDE5A (0.41) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9708165 0.91 ADORA3 (0.43) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9708763 0.91 PDE5A (0.43) AGTR1AGTR2PPARGKMT2A
SCHEMBL9708177 0.91 AGTR1 (0.39) AGTR1AGTR2PPARGKMT2APOLB
SCHEMBL9708180 0.91 AGTR1 (0.39) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9708572 0.91 ADORA3 (0.42) AGTR1AGTR2PPARGKMT2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed