SCHEMBL9707502

SCHEMBL9707502

CCn1c(=O)n(CCc2ccccc2)c(=O)c2c1nc(C(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.42
ADORA3 P0DMS8 3/20 0.41
SIRT1 Q96EB6 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41
SIRT5 Q9NXA8 1/20 0.41
AGTR1 P30556 3/20 0.41
AGTR2 P50052 1/20 0.40
PDE5A O76074 2/20 0.39
MAPT P10636 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707843 0.98 ADORA1 (0.42) ADORA1ADORA3AGTR1AGTR2PDE5A
SCHEMBL9708556 0.97 ADORA3 (0.42) ADORA1ADORA3AGTR1AGTR2MAPT
SCHEMBL9707601 0.95 ADORA3 (0.47) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9708001 0.95 ADORA3 (0.47) ADORA1ADORA3AGTR1AGTR2ADORA2A
SCHEMBL9708609 0.92 POLB (0.44) ADORA3MAPTCRHBPCRHR2NPSR1
SCHEMBL9707902 0.92 HPGD (0.43) AGTR1AGTR2MAPTCRHBPCRHR2
SCHEMBL9708021 0.92 ADORA3 (0.42) ADORA1ADORA3AGTR1ADORA2A
SCHEMBL9707419 0.92 ADORA3 (0.42) ADORA1ADORA3AGTR1ADORA2A
SCHEMBL9708350 0.90 ADORA3 (0.43) ADORA1ADORA3ADORA2A
SCHEMBL9708125 0.90 PDE5A (0.46) ADORA1ADORA3AGTR1AGTR2PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed