SCHEMBL9707419

SCHEMBL9707419

COCCn1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CCc2ccccc2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.42
ADORA2B P29275 5/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DCTPP1 Q9H773 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
USP1 O94782 2/20 0.38
ADORA1 P30542 1/20 0.38
AGTR1 P30556 2/20 0.38
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708021 1.00 ADORA3 (0.42) ADORA3ADORA2BALDH1A1LMNATSHR
SCHEMBL9707871 0.95 ADORA3 (0.42) ADORA3ADORA2BALDH1A1TSHRDCTPP1
SCHEMBL9708556 0.95 ADORA3 (0.42) ADORA3ADORA1AGTR1
SCHEMBL9707692 0.92 ADORA3 (0.40) ADORA3ADORA2BALDH1A1TSHRDCTPP1
SCHEMBL9707508 0.92 ADORA3 (0.42) ADORA3ADORA2BUSP1ADORA1ADORA2A
SCHEMBL9707777 0.92 ADORA3 (0.42) ADORA3ADORA2BUSP1ADORA1ADORA2A
SCHEMBL9707502 0.92 ADORA1 (0.42) ADORA3ADORA1AGTR1ADORA2A
SCHEMBL9708001 0.92 ADORA3 (0.47) ADORA3ADORA2BADORA1AGTR1ADORA2A
SCHEMBL9707745 0.92 ADORA2A (0.39) ADORA3ADORA2BALDH1A1TSHRDCTPP1
SCHEMBL9707601 0.92 ADORA3 (0.47) ADORA3ADORA2BADORA1AGTR1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed