SCHEMBL9707802

SCHEMBL9707802

CCCn1c(=O)n(CC(=O)OC)c(=O)c2c1nc(C(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
AGTR1 P30556 3/20 0.42
PPARG P37231 3/20 0.42
AGTR2 P50052 2/20 0.42
ADORA3 P0DMS8 4/20 0.39
ADORA1 P30542 2/20 0.39
MEN1 O00255 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 2/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707887 0.98 PPARG (0.41) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708112 0.95 KMT2A (0.42) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708371 0.95 KMT2A (0.44) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708822 0.93 KMT2A (0.40) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708179 0.93 KMT2A (0.42) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708471 0.93 KMT2A (0.43) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708309 0.93 KMT2A (0.40) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9707459 0.93 KMT2A (0.46) KMT2AAGTR1PPARGAGTR2MEN1
SCHEMBL9708440 0.91 AGTR1 (0.38) KMT2AAGTR1PPARGAGTR2ADORA3
SCHEMBL9708195 0.91 PPARG (0.39) KMT2AAGTR1PPARGAGTR2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed