SCHEMBL9708440

SCHEMBL9708440

COCCn1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CC(=O)OC)c1=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.38
AGTR2 P50052 2/20 0.38
PPARG P37231 2/20 0.38
KMT2A Q03164 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
ALDH1A1 P00352 2/20 0.37
USP1 O94782 4/20 0.36
MEN1 O00255 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.35
DCTPP1 Q9H773 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708822 0.98 KMT2A (0.40) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9708112 0.94 KMT2A (0.42) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9707887 0.94 PPARG (0.41) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9707871 0.93 ADORA3 (0.42) KMT2AADORA3ALDH1A1USP1MEN1
SCHEMBL9707917 0.92 KMT2A (0.41) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9708179 0.92 KMT2A (0.42) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9708195 0.91 PPARG (0.39) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9707802 0.91 KMT2A (0.42) AGTR1AGTR2PPARGKMT2AADORA3
SCHEMBL9707556 0.91 AGTR1 (0.40) AGTR1AGTR2PPARGKMT2AALDH1A1
SCHEMBL9708371 0.91 KMT2A (0.44) AGTR1AGTR2PPARGKMT2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed