SCHEMBL9707950

SCHEMBL9707950

CCCCCc1nc2c(c(=O)n(CCc3ccccc3)c(=O)n2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 8/20 0.48
AGTR2 P50052 8/20 0.48
USP2 O75604 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
POLB P06746 2/20 0.45
TP53 P04637 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.44
XBP1 P17861 1/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708599 0.98 AGTR1 (0.50) AGTR1AGTR2
SCHEMBL9707307 0.95 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL9708739 0.94 TSHR (0.45) AGTR1AGTR2ALDH1A1NPSR1POLB
SCHEMBL9708070 0.94 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL9708467 0.94 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL9707606 0.94 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL9708754 0.94 AGTR1 (0.48) AGTR1AGTR2USP2ALDH1A1NPSR1
SCHEMBL9707849 0.93 ADORA1 (0.51) AGTR1AGTR2
SCHEMBL9707432 0.93 AGTR1 (0.51) AGTR1AGTR2
SCHEMBL9707808 0.93 AGTR1 (0.49) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed