SCHEMBL9708739

SCHEMBL9708739

CCCc1nc2c(c(=O)n(CCc3ccccc3)c(=O)n2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
HSD17B10 Q99714 2/20 0.45
MAPT P10636 3/20 0.45
ALOX15 P16050 3/20 0.44
ALDH1A1 P00352 4/20 0.44
TP53 P04637 1/20 0.44
AGTR1 P30556 3/20 0.44
AGTR2 P50052 3/20 0.44
POLB P06746 1/20 0.44
HIF1A Q16665 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
HTT P42858 1/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708599 0.95 AGTR1 (0.50) AGTR1AGTR2
SCHEMBL9707950 0.94 AGTR1 (0.48) TSHRMAPTALDH1A1TP53AGTR1
SCHEMBL9708275 0.94 TSHR (0.46) TSHRHSD17B10MAPTALOX15ALDH1A1
SCHEMBL9708536 0.94 AGTR1 (0.46) HSD17B10MAPTALOX15AGTR1AGTR2
SCHEMBL9707867 0.94 ADORA3 (0.44) AGTR1AGTR2
SCHEMBL9708013 0.94 ADORA3 (0.44) AGTR1AGTR2
SCHEMBL9707576 0.94 TSHR (0.45) TSHRHSD17B10MAPTALOX15ALDH1A1
SCHEMBL9708848 0.93 ADORA1 (0.48) AGTR1AGTR2
SCHEMBL9707955 0.93 AGTR1 (0.46) HSD17B10MAPTALOX15AGTR1AGTR2
SCHEMBL9708134 0.92 ADORA1 (0.49) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed