SCHEMBL9708150

SCHEMBL9708150

CC(C)Cn1c(=O)n(-c2ccccc2)c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.36
AGTR2 P50052 1/20 0.36
ADORA1 P30542 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708473 0.94 ADORA3 (0.37) AGTR1AGTR2ADORA1ADORA3ADORA2A
SCHEMBL9707559 0.92 AGTR1 (0.41) AGTR1AGTR2ADORA1ADORA3
SCHEMBL9708413 0.92 AGTR1 (0.38) AGTR1AGTR2ADORA1ALDH1A1
SCHEMBL9708158 0.92 ADORA3 (0.41) AGTR1AGTR2ADORA1ADORA3PDE1A
SCHEMBL9708540 0.91 AGTR1 (0.38) AGTR1AGTR2ALDH1A1
SCHEMBL9707998 0.90 AGTR1 (0.39) AGTR1AGTR2ADORA1ADORA3ADORA2A
SCHEMBL9708206 0.90 AGTR1 (0.42) AGTR1AGTR2
SCHEMBL9709079 0.90 PDE1A (0.43) PDE1APDE1BPDE1CALDH1A1
SCHEMBL9708630 0.90 AGTR1 (0.39) AGTR1AGTR2ALDH1A1
SCHEMBL9708074 0.89 ADORA1 (0.38) AGTR1AGTR2ADORA1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed