SCHEMBL9708328

SCHEMBL9708328

CCn1c(=O)n(C(C)c2ccccc2)c(=O)c2c1nc(C1CCCCC1)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 5/20 0.40
KMT2A Q03164 1/20 0.40
AGTR1 P30556 5/20 0.38
AGTR2 P50052 4/20 0.38
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708020 0.94 ADORA3 (0.42) PDE5AKMT2AAGTR1AGTR2ADORA3
SCHEMBL9708034 0.94 PDE5A (0.40) PDE5AKMT2AAGTR1AGTR2ADORA3
SCHEMBL9708670 0.94 KMT2A (0.40) KMT2AAGTR1AGTR2
SCHEMBL9708680 0.92 KMT2A (0.42) PDE5AKMT2AAGTR1AGTR2ADORA3
SCHEMBL9708207 0.92 KMT2A (0.42) KMT2AAGTR1AGTR2
SCHEMBL9707827 0.91 AGTR1 (0.38) KMT2AAGTR1AGTR2
SCHEMBL9707991 0.91 AGTR1 (0.38) KMT2AAGTR1AGTR2
SCHEMBL9708118 0.91 PDE5A (0.39) PDE5AKMT2AAGTR1AGTR2
SCHEMBL9707993 0.90 ADORA3 (0.42) KMT2AAGTR1AGTR2ADORA3
SCHEMBL9708842 0.90 PPARG (0.38) KMT2AAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed