SCHEMBL9709849

SCHEMBL9709849

Cc1cc(NCc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CD38 P28907 8/20 0.47
CYP3A4 P08684 2/20 0.47
AGTR1 P30556 4/20 0.45
AGTR2 P50052 4/20 0.45
KCNH2 Q12809 1/20 0.43
USP1 O94782 6/20 0.41
WDR48 Q8TAF3 6/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709642 0.89 AGTR1 (0.48) CD38CYP3A4AGTR1AGTR2KCNH2
SCHEMBL9709806 0.86 AGTR1 (0.46) CD38CYP3A4AGTR1AGTR2
SCHEMBL3051876 0.86 CD38 (0.46) CD38AGTR1AGTR2
SCHEMBL9709829 0.86 AGTR1 (0.47) CD38AGTR1AGTR2USP1WDR48
SCHEMBL9709754 0.84 AGTR1 (0.47) CD38AGTR1AGTR2
SCHEMBL3058746 0.84 AGTR1 (0.50) AGTR1AGTR2
SCHEMBL9710150 0.80 TLR7 (0.47) AGTR1AGTR2USP1WDR48
SCHEMBL9704665 0.79 AGTR1 (0.70) AGTR1AGTR2
SCHEMBL9710179 0.79 AGTR1 (0.47) CD38AGTR1AGTR2
SCHEMBL9464440 0.78 AGTR1 (0.70) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO claimed
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO disclosed