SCHEMBL9710088

SCHEMBL9710088

Clc1ccc(CCNCCN2CCCC2)cc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 17/20 1.00
SMYD2 Q9NRG4 3/20 0.62
TP53 P04637 2/20 0.58
CYP1A2 P05177 2/20 0.58
CYP2D6 P10635 2/20 0.58
TSHR P16473 2/20 0.58
GRIN2D O15399 1/20 0.57
GRIN3B O60391 1/20 0.57
CYP3A4 P08684 1/20 0.57
GRIN1 Q05586 1/20 0.57
GRIN2A Q12879 1/20 0.57
GRIN2B Q13224 1/20 0.57
GRIN2C Q14957 1/20 0.57
GRIN3A Q8TCU5 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756580 0.85 SIGMAR1 (0.74) SIGMAR1SMYD2TP53CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL5757385 0.85 SIGMAR1 (0.74) SIGMAR1TP53CYP1A2CYP2D6TSHR
Hydrochloric Acid SCHEMBL5754393 0.84 SIGMAR1 (0.72) SIGMAR1SMYD2TP53CYP1A2CYP2D6
SCHEMBL16511553 0.84 SIGMAR1 (0.83) SIGMAR1
SCHEMBL5804316 0.82 SIGMAR1 (0.93) SIGMAR1TP53CYP1A2CYP2D6TSHR
SCHEMBL16511184 0.82 SIGMAR1 (0.80) SIGMAR1CYP1A2CYP3A4
SCHEMBL27550763 0.80 SIGMAR1 (0.65) SIGMAR1SMYD2
SCHEMBL6961777 0.80 SIGMAR1 (0.76) SIGMAR1TP53CYP1A2CYP2D6TSHR
SCHEMBL17476322 0.79 SMYD2 (1.00) SIGMAR1SMYD2TP53CYP1A2CYP2D6
SCHEMBL9019137 0.76 SIGMAR1 (1.00) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210379016-A1 THERAPEUTICS AND METHODS OF TREATMENT OF ANGIOTENSIN-CONVERTING ENZYME 2 ASSOCIATED CONDITIONS BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL COLLEGE (US) 2021-12-09 US disclosed
WO-1992022279-A2 N-[ARYLETHYL]-N-ALKYL-2-(1-PYRROLIDINYL)ETHYLAMINE DERIVATIVES FOR CNS DISORDERS G.D. SEARLE & CO. (US) 1992-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210379016-A1 THERAPEUTICS AND METHODS OF TREATMENT OF ANGIOTENSIN-CONVERTING ENZYME 2 ASSOCIATED CONDITIONS ACE2, ACE, AGTR2 SIGMAR1 10/4885SMYD2 3068/4885TP53 3983/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.