SCHEMBL9710583

SCHEMBL9710583

OC(c1ccccc1)[C@H]1CN(CCc2ccccc2)CC[C@]1(O)c1ccccc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.78
ALDH1A1 P00352 2/20 0.78
KDM4E B2RXH2 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
SLC6A3 Q01959 1/20 0.49
OPRM1 P35372 5/20 0.46
OPRK1 P41145 3/20 0.46
OPRD1 P41143 2/20 0.46
ARRB1 P49407 1/20 0.46
OPRL1 P41146 3/20 0.45
SIGMAR1 Q99720 1/20 0.45
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9297947 0.92 TSHR (0.73) TSHRALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL11867116 0.88 ALDH1A1 (1.00) TSHRALDH1A1KDM4ESLC6A3OPRM1
SCHEMBL11870408 0.87 ALDH1A1 (0.72) TSHRALDH1A1KDM4ECYP1A2CYP3A4
SCHEMBL9710602 0.87 ALDH1A1 (0.72) TSHRALDH1A1SLC6A3OPRM1OPRL1
SCHEMBL9173912 0.86 ALDH1A1 (0.71) TSHRALDH1A1SLC6A3OPRM1OPRL1
SCHEMBL9711021 0.85 ALDH1A1 (0.64) TSHRALDH1A1HTR2ASLC6A3SIGMAR1
SCHEMBL11872237 0.84 ALDH1A1 (0.68) TSHRALDH1A1SLC6A3OPRM1OPRK1
SCHEMBL11867863 0.84 ALDH1A1 (0.68) TSHRALDH1A1SLC6A3OPRM1OPRK1
SCHEMBL11861506 0.84 ALDH1A1 (0.68) TSHRALDH1A1SLC6A3OPRM1OPRK1
SCHEMBL9296560 0.83 ALDH1A1 (0.74) TSHRALDH1A1KDM4ESLC6A3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992018480-A1 1,3,4-TRISUBSTITUTED PIPERIDINE DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1992-10-29 WO disclosed