SCHEMBL9712834

SCHEMBL9712834

CCCCOc1ccc(C#Cc2ccc(OC(F)(F)C(F)F)cc2)nc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACACB O00763 10/20 0.48
MCHR1 Q99705 7/20 0.43
CYP2D6 P10635 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP19A1 P11511 1/20 0.39
CYP2C19 P33261 1/20 0.39
CHRM1 P11229 2/20 0.39
HTR2A P28223 2/20 0.39
CYP3A4 P08684 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713534 0.98 ACACB (0.47) ACACBMCHR1CYP2D6CYP2C9CYP1A2
SCHEMBL9713338 0.96 ACACB (0.46) ACACBMCHR1CYP2D6CYP2C9CYP1A2
SCHEMBL9713638 0.96 ACACB (0.46) ACACBMCHR1CYP2D6CYP2C9CYP1A2
SCHEMBL9712812 0.96 ACACB (0.46) ACACBMCHR1CYP2D6CYP2C9CYP1A2
SCHEMBL10524909 0.95 ACACB (0.50) ACACBMCHR1CYP2D6CYP2C9CYP1A2
SCHEMBL9712880 0.95 ACACB (0.53) ACACBMCHR1CHRM1HTR2A
SCHEMBL9713556 0.90 ACACB (0.52) ACACBMCHR1
SCHEMBL9713293 0.89 ACACB (0.51) ACACBMCHR1CYP2D6CYP2C9CYP1A2
SCHEMBL9713252 0.87 ACACB (0.47) ACACBMCHR1CYP1A2CYP3A4KDM4E
SCHEMBL9713057 0.86 ACACB (0.49) ACACBMCHR1CYP2D6CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164114-A LIQUID CRYSTAL MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1992-11-17 US disclosed
EP-0306521-B1 ETHINE DERIVATIVES AS COMPOUNDS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1991-10-16 EP disclosed