SCHEMBL9713841

SCHEMBL9713841

CCOC(=O)COc1cc(N)ccc1S(=O)(=O)c1ccc(N)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.56
GAA P10253 1/20 0.56
MAPK1 P28482 2/20 0.47
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 4/20 0.40
CASP3 P42574 1/20 0.39
CASP7 P55210 1/20 0.39
CASP9 P55211 1/20 0.39
LMNA P02545 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
MAOA P21397 1/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
CYP2C9 P11712 1/20 0.39
NTSR1 P30989 1/20 0.39
CYP2C19 P33261 1/20 0.39
USP2 O75604 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714211 0.84 ALDH1A1 (0.41) NPSR1GAAMAPK1POLBSMN1; SMN2
SCHEMBL9713926 0.83 ALDH1A1 (0.50) GAAALDH1A1LMNACYP3A4HPGD
SCHEMBL13215154 0.77 MAPK1 (0.56) NPSR1GAAMAPK1POLBSMN1; SMN2
SCHEMBL13215132 0.76 MAPK1 (0.52) NPSR1GAAMAPK1ALDH1A1CASP3
SCHEMBL31384765 0.76 MAPK1 (0.52) NPSR1GAAMAPK1ALDH1A1CASP3
SCHEMBL3533533 0.76 ALDH1A1 (0.65) GAAMAPK1ALDH1A1CYP1A2MAPT
SCHEMBL2839402 0.76 ALDH1A1 (0.58) GAAMAPK1ALDH1A1CASP3CASP7
SCHEMBL4861445 0.76 MAPK1 (0.57) NPSR1GAAMAPK1POLBSMN1; SMN2
SCHEMBL4861358 0.73 MAPK1 (0.55) NPSR1GAAMAPK1POLBALDH1A1
SCHEMBL3531540 0.73 ALDH1A1 (0.56) NPSR1GAAMAPK1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed