SCHEMBL9714211

SCHEMBL9714211

CN(C)C(=O)COc1cc(N)ccc1S(=O)(=O)c1ccc(N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR6 P50406 3/20 0.38
HSD11B1 P28845 1/20 0.38
LMNA P02545 1/20 0.38
MPO P05164 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
POLB P06746 1/20 0.37
PKM P14618 2/20 0.37
CYP2C19 P33261 1/20 0.37
HKDC1 Q2TB90 1/20 0.36
RAPGEF3 O95398 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713926 0.84 ALDH1A1 (0.50) ALDH1A1HTR6HSD11B1LMNAMPO
SCHEMBL9713841 0.84 NPSR1 (0.56) ALDH1A1SMN1; SMN2NPSR1MAPK1LMNA
SCHEMBL7777372 0.72 MEN1 (0.51) ALDH1A1SMN1; SMN2NPSR1MEN1MAPK1
SCHEMBL15651103 0.72 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2NPSR1MEN1MAPK1
SCHEMBL8320409 0.71 SMN1; SMN2 (0.65) ALDH1A1SMN1; SMN2MAPK1TSHRPOLB
SCHEMBL21305523 0.70 SMN1; SMN2 (0.59) ALDH1A1SMN1; SMN2NPSR1MEN1MAPK1
SCHEMBL9713990 0.68 HTR6 (0.50) ALDH1A1MEN1KMT2AHTR6HSD11B1
SCHEMBL3928072 0.68 CYP19A1 (0.55) ALDH1A1SMN1; SMN2HTR6PKMKDM4E
SCHEMBL9713812 0.67 PKM (0.49) ALDH1A1SMN1; SMN2MEN1KMT2AHTR6
SCHEMBL157598 0.67 HSD17B10 (0.59) ALDH1A1SMN1; SMN2MEN1MAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed