SCHEMBL9713981

SCHEMBL9713981

CC1(C)CCC(C)(C)c2cc(C#Cc3ccc(C(=O)O)cc3)c(F)cc21

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARB P10826 14/20 0.69
RARG P13631 14/20 0.69
RARA P10276 9/20 0.69
CYP26A1 O43174 1/20 0.69
CYP3A4 P08684 1/20 0.69
CRABP2 P29373 1/20 0.69
RXRA P19793 12/20 0.60
RXRB P28702 9/20 0.51
RXRG P48443 7/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9483542 0.85 RARB (0.71) RARBRARGRARACYP26A1CYP3A4
SCHEMBL31756435 0.84 RARB (0.72) RARBRARGRARACYP26A1CYP3A4
SCHEMBL22410909 0.84 RARB (0.72) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9487042 0.83 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8460052 0.82 RARB (0.70) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9484944 0.82 RARB (0.43) RARBRARGRARACYP26A1CYP3A4
SCHEMBL3302926 0.82 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL29353973 0.82 RARB (1.00) RARBRARGRARACYP26A1CYP3A4
SCHEMBL24410702 0.80 RXRA (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5084011 0.77 RARB (0.63) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5126371-A Precancerous skin conditions, acne, psoriasis BASF AKTEINGESELLSCHAFT (DE) 1992-06-30 US disclosed
US-4994489-A Ester derivatives of diarylacetylenes, their compositions and their use in acne treatment BASF AKTIENGESELLSCHAFT 1991-02-19 US disclosed
US-4806558-A Diarylacetylenes and their use in treating acne BASF AKTIENGESELLSCHAFT (DE) 1989-02-21 US disclosed