SCHEMBL9714878

SCHEMBL9714878

CC(=O)C(C)(C)C(Cl)/C=C(/Cl)c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.41
TRPA1 O75762 3/20 0.38
GAA P10253 1/20 0.38
CES2 O00748 2/20 0.37
CES1 P23141 2/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.36
ELANE P08246 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
MEN1 O00255 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714881 1.00 POLB (0.41) POLBTRPA1GAACES2CES1
SCHEMBL9774843 0.84 TSHR (0.41) TSHRMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL9774831 0.84 TSHR (0.41) TSHRMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL9774839 0.84 TSHR (0.41) TSHRMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL9714880 0.84 GSK3B (0.41) POLBTRPA1GAACES2CES1
SCHEMBL9714877 0.84 GSK3B (0.41) POLBTRPA1GAACES2CES1
SCHEMBL9714886 0.82 GSK3B (0.42) POLBTRPA1GAACES2CES1
SCHEMBL9714887 0.82 GSK3B (0.42) POLBTRPA1GAACES2CES1
SCHEMBL11472847 0.76 POLB (0.36) POLBTRPA1GAAMAPK1TSHR
SCHEMBL11068444 0.75 PTGS2 (0.40) POLBTRPA1MAPK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0323625-B1 Process for preparing 3-[2-chloro-2(4-chlorophenyl)-vinyl]-2,2-dimethyl-cyclopropane carboxylic acid BAYER AG (DE) 1992-09-09 EP disclosed
US-4992577-A Preparation of 3-vinyl-substituted 2,2-dimethylcyclopropane-1-carboxylic acids and esters and intermediates therefor BAYER AKTIENGESELLSCHAFT (DE) 1991-02-12 US disclosed
US-4897505-A Process for the preparation of 3-(2-chloro-2-(4-chloro-phenyl)-vinyl)-2,2-dimethylcyclopropanecarboxylic acid BAYER AKTIENGESELLSCHAFT (DE) 1990-01-30 US disclosed
EP-0323625-A2 Process for preparing 3-[2-chloro-2(4-chlorophenyl)-vinyl]-2,2-dimethyl-cyclopropane carboxylic acid BAYER AG (DE) 1989-07-12 EP disclosed
EP-0095047-B1 PROCESS FOR THE PREPARATION OF 3-VINYL-SUBSTITUTED 2,2-DIMETHYL-CYCLOPROPANE-1-CARBOXYLIC ACIDS OR THEIR ESTERS, AND INTERMEDIATE PRODUCTS THEREFOR BAYER AG (DE) 1985-11-27 EP disclosed
EP-0095047-A1 Process for the preparation of 3-vinyl-substituted 2,2-dimethyl-cyclopropane-1-carboxylic acids or their esters, and intermediate products therefor BAYER AG (DE) 1983-11-30 EP disclosed