SCHEMBL9718255

SCHEMBL9718255

N#C/C=C/Cc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.61
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
ARG2 P78540 1/20 0.47
ALDH1A1 P00352 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
MAPK1 P28482 1/20 0.40
TOP1 P11387 1/20 0.39
TSHR P16473 1/20 0.39
MAOA P21397 2/20 0.37
CALM1 P0DP23 1/20 0.36
ATP4A P20648 1/20 0.35
ATP4B P51164 1/20 0.35
IDO1 P14902 2/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
KCNH2 Q12809 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10563302 1.00 MAOB (0.61) MAOBCA1CA2ARG2ALDH1A1
SCHEMBL3804445 0.79 CYP1A1 (0.38) MAOBALDH1A1CYP1A1CYP1A2CYP1B1
SCHEMBL10539962 0.78 GPR52 (0.46) MAOBALDH1A1
SCHEMBL10539956 0.78 GPR52 (0.46) MAOBALDH1A1
SCHEMBL28684461 0.78 MAOB (0.41) MAOBALDH1A1CYP1A2MAPK1TSHR
SCHEMBL17050914 0.78 MAOB (0.40) MAOBALDH1A1CYP1A1CYP1A2CYP1B1
SCHEMBL145088 0.77 MAOB (0.61) MAOBCA1CA2ARG2MAPK1
SCHEMBL334261 0.77 MAOB (0.61) MAOBCA1CA2ARG2MAPK1
SCHEMBL261253 0.77 MAOB (0.61) MAOBCA1CA2ARG2MAPK1
SCHEMBL155054 0.77 MAOB (1.00) MAOBCA1CA2ARG2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4136077-A REACTION PRODUCT OF OLEFINICALLY-UNSATURATED NITRILE AND A MONOOLEFINIC HYDROCARBON AS PLASTICIZER FOR CONJUGATED DIENE-UNSATURATED NITRILE RUBBER PHILLIPS PETROLEUM COMPANY (US) 1979-01-23 US claimed
EP-0463402-A2 Ethylene polymers or copolymers having improved insulating properties, compositions, and power cables made therefrom NIPPON PETROCHEMICALS COMPANY, LIMITED (JP) 1992-01-02 EP disclosed
US-4472319-A Preparation of unsaturated nitriles using a surfactant PHILLIPS PETROLEUM COMPANY (US) 1984-09-18 US disclosed
US-4288626-A CATALYTIC, PRETREATMENT OF FEED WITH CRYSTALLINE ZEOLITE PHILLIPS PETROLEUM COMPANY (US) 1981-09-08 US disclosed
US-4275237-A ETHYLENICALLY UNSATURATED POLYAMINE CURING AGENTS PHILIPS PETROLEUM COMPANY (US) 1981-06-23 US disclosed
US-4255352-A TANK REACTORS IN SERIES PHILLIPS PETROLEUM COMPANY (US) 1981-03-10 US disclosed
US-4243769-A NITRILE POLYMER, HYDROXY OR ESTER POLYMER, ACID NATIONAL DISTILLERS AND CHEMICAL CORP. (US) 1981-01-06 US disclosed
US-4217303-A UNSATURATED HYDROCARBON, ADDUCT, UNSATURATED DINITRILE, BY-PRODUCT INHIBITION PHILLIPS PETROLEUM COMPANY (US) 1980-08-12 US disclosed
US-4200586-A Inhibiting the carbon-carbon double bond isomerization of substituted or unsubstituted hydrocarbon compounds PHILLIPS PETROLEUM COMPANY (US) 1980-04-29 US disclosed
US-4195155-A Hydrogenated polynitrile mixture and use as epoxy hardener PHILLIPS PETROLEUM COMPANY (US) 1980-03-25 US disclosed
US-4136077-A REACTION PRODUCT OF OLEFINICALLY-UNSATURATED NITRILE AND A MONOOLEFINIC HYDROCARBON AS PLASTICIZER FOR CONJUGATED DIENE-UNSATURATED NITRILE RUBBER PHILLIPS PETROLEUM COMPANY (US) 1979-01-23 US disclosed
US-4117001-A TO RECOVER STARTING MATERIALS PHILLIPS PETROLEUM COMPANY (US) 1978-09-26 US disclosed
US-4117002-A PYROLYSIS OF HEAVIES FORMED IN PRODUCTION OF UNSATURATED DINITRILES PHILLIPS PETROLEUM COMPANY (US) 1978-09-26 US disclosed
US-3985786-A REACTING AN OLEFINICALLY UNSATURATED NITRILE, AN OLEFINIC HYDROCARBON AND THEIR MONOADDUCT IN WATER PHILLIPS PETROLEUM COMPANY (US) 1976-10-12 US disclosed