SCHEMBL9718295

SCHEMBL9718295

CC(C)(Cc1ccc(F)cc1)NC(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
MMP2 P08253 1/20 0.49
MMP8 P22894 1/20 0.49
MMP12 P39900 1/20 0.49
ADAMTS5 Q9UNA0 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HPGD P15428 2/20 0.46
DPP4 P27487 1/20 0.45
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 2/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RIPK1 Q13546 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8384266 0.86 KDM4E (0.53) KDM4EMMP2MMP8MMP12ADAMTS5
SCHEMBL4171208 0.84 ESR1 (0.59) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL27461036 0.84 CYP3A4 (0.50) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL5948337 0.83 CYP3A4 (0.67) MMP8ALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL25344198 0.83 MMP2 (0.51) KDM4EMMP2MMP8MMP12ADAMTS5
SCHEMBL14185300 0.83 KDM4E (0.62) KDM4EMMP2MMP8MMP12ADAMTS5
SCHEMBL7906601 0.83 KDM4E (0.50) KDM4EMMP2MMP8MMP12ADAMTS5
SCHEMBL16041240 0.82 ALDH1A1 (0.49) ALDH1A1CYP3A4CYP2C9CYP2C19HPGD
SCHEMBL1998840 0.82 CYP3A4 (0.49) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL28794058 0.82 CYP2C9 (0.49) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5153327-A 7-Oxabicycloheptyl substituted heterocyclic amide or ester prostaglandin analogs useful in the treatment of thrombotic and vasospastic disease E. R. SQUIBB & SONS, INC. (US) 1992-10-06 US disclosed
US-5100889-A Thromboxane A2 receptor antagonists, thromboxane synthetase inhibitor E. R. SQUIBB & SONS, INC. (US) 1992-03-31 US disclosed