SCHEMBL9719084

SCHEMBL9719084

CCOC(=O)C(C#N)c1cc(OC)c(OC)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
KDM4E B2RXH2 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
GAA P10253 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPK1 P28482 1/20 0.43
FNTA P49354 1/20 0.43
FNTB P49356 1/20 0.43
HPGD P15428 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744359 0.84 ALDH1A1 (0.51) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL9719027 0.83 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL15475932 0.82 KMT2A (0.47) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL9719048 0.81 SMN1; SMN2 (0.38) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL10040724 0.80 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL491076 0.78 ALDH1A1 (0.53) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL17466005 0.77 MEN1 (0.58) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL11436992 0.77 KMT2A (0.46) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL22995348 0.77 KMT2A (0.58) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL3458704 0.77 ALDH1A1 (0.51) ALDH1A1KMT2AMEN1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132463-A Cardiovascular, skin, kidney, respiratory system, and gastrointestinal disorders MERCK & CO., INC. (US) 1992-07-21 US disclosed
EP-0257921-B1 NEW 1,3-DIARYL CYCLOPENTANES AND DERIVATIVES THEREOF AS PAF ANTAGONISTS MERCK & CO. INC. (US) 1992-04-15 EP disclosed
US-5047420-A Platelet activating factor MERCK & CO., INC. (US) 1991-09-10 US disclosed
EP-0257921-A2 New 1,3-diaryl cyclopentanes and derivatives thereof as paf antagonists MERCK & CO. INC. (US) 1988-03-02 EP disclosed