SCHEMBL9720106

SCHEMBL9720106

Fc1ccc(C2(Br)C=CC=CC2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.36
SLC6A4 P31645 5/20 0.36
SLC6A2 P23975 5/20 0.33
CHRNA1 P02708 1/20 0.31
CHRNG P07510 1/20 0.31
CHRNB1 P11230 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
CHRND Q07001 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720104 0.75 SLC6A3 (0.35) SLC6A3SLC6A4SLC6A2CHRNA1CHRNG
SCHEMBL5177413 0.74 CYP2A6 (0.32)
SCHEMBL276639 0.72 HDAC4 (0.32)
SCHEMBL8971076 0.66 SLC6A2 (0.33) SLC6A3SLC6A4SLC6A2
SCHEMBL25599865 0.63 ALDH1A1 (0.37)
SCHEMBL9230201 0.63 SLC6A3 (0.40) SLC6A3SLC6A4SLC6A2CHRNA1CHRNG
SCHEMBL30773513 0.62 SLC6A3 (0.46) SLC6A3SLC6A4SLC6A2CHRNA1CHRNG
SCHEMBL5865741 0.62 KDM1A (0.31)
SCHEMBL5187900 0.60 HDAC4 (0.33) SLC6A4
SCHEMBL27955335 0.59 SLC6A3 (0.44) SLC6A3SLC6A4SLC6A2CHRNA1CHRNG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0338054-B1 CROSS COUPLING OF TITANIUM ORGANYLS MERCK PATENT GmbH (DE) 1992-12-30 EP disclosed
EP-0338054-A1 CROSS COUPLING OF TITANIUM ORGANYLS MERCK PATENT GmbH (DE) 1989-10-25 EP disclosed
WO-1989003812-A1 CROSS COUPLING OF TITANIUM ORGANYLS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-05-05 WO disclosed