SCHEMBL9720258

SCHEMBL9720258

CCCCCCCCCCCCCCCCCCOCC(COCCCc1cccnc1)Oc1ncccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HRH1 P35367 2/20 0.41
LMNA P02545 2/20 0.40
CYP2A6 P11509 1/20 0.40
TLR2 O60603 1/20 0.39
NFKB1 P19838 2/20 0.39
NFKB2 Q00653 2/20 0.39
RELA Q04206 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TRPV1 Q8NER1 1/20 0.38
TBXAS1 P24557 2/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720249 0.83 TDP1 (0.60) TDP1L3MBTL1HRH1LMNACYP2A6
SCHEMBL10061567 0.77 L3MBTL1 (0.75) TDP1L3MBTL1HRH1CYP2A6CYP3A4
SCHEMBL2098501 0.76 TDP1 (0.55) TDP1L3MBTL1HRH1CYP2A6TBXAS1
SCHEMBL23015074 0.76 TDP1 (0.68) TDP1L3MBTL1HRH1CYP2A6TRPV1
SCHEMBL2608878 0.76 TDP1 (0.54) TDP1L3MBTL1HRH1CYP2A6CYP3A4
SCHEMBL10385452 0.75 MEN1 (0.54) LMNACYP3A4MAPTSMN1; SMN2PLA2G2A
SCHEMBL9720214 0.75 MEN1 (0.54) LMNACYP3A4MAPTSMN1; SMN2PLA2G2A
SCHEMBL25380936 0.75 TDP1 (0.96) TDP1L3MBTL1HRH1CYP2A6TRPV1
SCHEMBL6114843 0.75 TDP1 (0.96) TDP1L3MBTL1HRH1CYP2A6TRPV1
SCHEMBL25381701 0.75 TDP1 (0.96) TDP1L3MBTL1HRH1CYP2A6TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081245-A Selective antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-01-14 US disclosed
EP-0356765-A2 Carboxylic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-03-07 EP disclosed