SCHEMBL9720299

SCHEMBL9720299

CCCCC=C(C)c1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 3/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
NAAA Q02083 1/20 0.42
LMNA P02545 3/20 0.39
NPC1 O15118 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 2/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.35
STAT3 P40763 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1053053 0.81 TBXAS1 (0.45) TBXAS1NAAACYP3A4CYP1A2CYP2C9
SCHEMBL1053054 0.81 TBXAS1 (0.45) TBXAS1NAAACYP3A4CYP1A2CYP2C9
SCHEMBL21462939 0.81 TBXAS1 (0.45) TBXAS1NAAACYP3A4CYP1A2CYP2C9
SCHEMBL20708210 0.80 L3MBTL1 (0.39) HDAC3HDAC1HDAC2NAAACYP3A4
SCHEMBL9720318 0.80 TBXAS1 (0.68) TBXAS1HDAC3HDAC1HDAC2LMNA
SCHEMBL2566604 0.79 HSD17B3 (0.47) TBXAS1LMNACYP3A4CYP2D6CYP1A2
SCHEMBL2566602 0.79 HSD17B3 (0.47) TBXAS1LMNACYP3A4CYP2D6CYP1A2
SCHEMBL2768533 0.76 TBXAS1 (0.48) TBXAS1NAAA
SCHEMBL2768526 0.76 TBXAS1 (0.48) TBXAS1NAAA
SCHEMBL2768530 0.76 TBXAS1 (0.48) TBXAS1NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5148817-A Heterocyclic hydroxy-substituted carboxylic compound as flavor additive PHILIP MORRIS INCORPORATED (US) 1992-09-22 US claimed
US-5148817-A Heterocyclic hydroxy-substituted carboxylic compound as flavor additive PHILIP MORRIS INCORPORATED (US) 1992-09-22 US disclosed
US-4592373-A Smoking compositions PHILIP MORRIS INC. (US) 1986-06-03 US disclosed
EP-0052969-A2 Flavorant compounds, their pyrolysis products, and smoking and food compositions containing them PHILIP MORRIS INCORPORATED (US) 1982-06-02 EP disclosed