SCHEMBL9720583

SCHEMBL9720583

C=Cc1cccc(C(=O)CC)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.46
TP53 P04637 1/20 0.46
KDM4E B2RXH2 1/20 0.43
MAPT P10636 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
UNG P13051 1/20 0.42
PTGS2 P35354 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
ATM Q13315 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
GAA P10253 1/20 0.39
TTR P02766 2/20 0.37
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8580569 0.85 MAPT (0.44) TDP1KDM4EMAPTSMN1; SMN2L3MBTL1
SCHEMBL3033625 0.84 MAPT (0.43) TDP1KDM4EMAPTSMN1; SMN2L3MBTL1
SCHEMBL25031282 0.82 GSK3B (0.52) TDP1TP53UNGPTGS2TTR
SCHEMBL29838127 0.82 ALDH1A1 (0.52) TDP1TP53KDM4EUNGPTGS2
SCHEMBL25031506 0.82 ALDH1A1 (0.52) TDP1TP53KDM4EUNGPTGS2
SCHEMBL29838103 0.82 GSK3B (0.52) TDP1TP53UNGPTGS2TTR
SCHEMBL4443836 0.81 CYP2D6 (0.45) TDP1TP53UNGPTGS2MEN1
SCHEMBL1720943 0.81 MEN1 (0.59) TDP1TP53KDM4EMAPTSMN1; SMN2
SCHEMBL10389972 0.80 SMN1; SMN2 (0.54) TDP1MAPTSMN1; SMN2L3MBTL1ALDH1A1
SCHEMBL14992845 0.80 TDP1 (0.47) TDP1TP53MAPTSMN1; SMN2UNG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed