SCHEMBL9720608

SCHEMBL9720608

Cc1cccc(C(=O)C(C)CN2CCCC2)c1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.56
ADRA2B P18089 2/20 0.56
DRD3 P35462 2/20 0.56
SIGMAR1 Q99720 2/20 0.56
HRH3 Q9Y5N1 2/20 0.56
ALDH1A1 P00352 3/20 0.55
LMNA P02545 2/20 0.55
CYP2D6 P10635 1/20 0.50
ADRA2C P18825 1/20 0.50
CHRM3 P20309 1/20 0.50
OPRD1 P41143 1/20 0.50
KCNH2 Q12809 1/20 0.50
FNTA P49354 1/20 0.49
FNTB P49356 1/20 0.49
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MITF O75030 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9720679 0.99 ALDH1A1 (0.57) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL13304408 0.87 CHRM2 (0.61) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL4936216 0.87 CHRM2 (0.61) CHRM2ADRA2BDRD3SIGMAR1HRH3
Hydrochloric Acid SCHEMBL30463042 0.86 ALDH1A1 (0.62) CHRM2ADRA2BDRD3SIGMAR1HRH3
Hydrochloric Acid SCHEMBL30463043 0.86 ALDH1A1 (0.62) CHRM2ADRA2BDRD3SIGMAR1HRH3
Hydrochloric Acid SCHEMBL3339536 0.86 ALDH1A1 (0.62) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL10706138 0.80 HRH3 (0.52) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL10852083 0.80 CHRM2 (0.53) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL10707183 0.79 HRH3 (0.55) CHRM2ADRA2BDRD3SIGMAR1HRH3
SCHEMBL10859044 0.78 CHRM2 (0.57) CHRM2ADRA2BDRD3SIGMAR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP claimed
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed