SCHEMBL9720946

SCHEMBL9720946

CC(C)CN(CCCC(O)(c1ccccc1)c1ccccc1F)CC(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.48
CHRM4 P08173 5/20 0.46
CHRM5 P08912 5/20 0.46
CHRM3 P20309 5/20 0.46
CHRM2 P08172 4/20 0.46
CHRM1 P11229 4/20 0.46
BCL2 P10415 3/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
ADRA1A P35348 1/20 0.45
OPRK1 P41145 1/20 0.45
KCNH2 Q12809 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.42
LMNA P02545 1/20 0.38
ALDH1A1 P00352 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KCNN4 O15554 2/20 0.35
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9716797 0.92 SIGMAR1 (0.39) SIGMAR1CHRM4CHRM5CHRM3CHRM2
SCHEMBL9716801 0.86 SIGMAR1 (0.62) SIGMAR1CHRM4CHRM5CHRM3CHRM2
Hydrochloric Acid SCHEMBL9716825 0.85 CHRM4 (0.62) SIGMAR1CHRM4CHRM5CHRM3CHRM2
SCHEMBL9716891 0.85 HTR2A (0.65) SIGMAR1CHRM4CHRM5CHRM3CHRM2
SCHEMBL9716774 0.80 SIGMAR1 (0.55) SIGMAR1CHRM4CHRM5CHRM3CHRM2
Maleic Acid SCHEMBL9716787 0.78 SIGMAR1 (0.52) SIGMAR1CHRM4CHRM5CHRM3CHRM2
Fumaric Acid SCHEMBL9716792 0.78 SIGMAR1 (0.52) SIGMAR1CHRM4CHRM5CHRM3CHRM2
Maleic Acid SCHEMBL9716806 0.77 BCL2 (0.46) SIGMAR1CHRM4CHRM5CHRM3CHRM2
Fumaric Acid SCHEMBL9716813 0.77 BCL2 (0.46) SIGMAR1CHRM4CHRM5CHRM3CHRM2
SCHEMBL9716807 0.76 HTR2A (0.52) SIGMAR1CHRM4CHRM5CHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5089529-A Antiarrhythmia agents NIPPON SHINYAKU CO., LTD. (JP) 1992-02-18 US claimed
US-5089529-A Antiarrhythmia agents NIPPON SHINYAKU CO., LTD. (JP) 1992-02-18 US disclosed