SCHEMBL9722386

SCHEMBL9722386

CCCc1cc2c(cc1O)C(C)(C)C(C)(C)O2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.41
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
TRPA1 O75762 2/20 0.35
CNR1 P21554 2/20 0.35
CNR2 P34972 2/20 0.35
TRPV1 Q8NER1 2/20 0.35
TRPV3 Q8NET8 2/20 0.35
TRPV4 Q9HBA0 2/20 0.35
TRPV2 Q9Y5S1 2/20 0.35
ALOX5 P09917 1/20 0.33
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
XBP1 P17861 1/20 0.32
HIF1A Q16665 1/20 0.32
PTPN1 P18031 1/20 0.32
PTPN11 Q06124 1/20 0.32
TYR P14679 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15257370 0.76 RXRA (0.38) ALDH1A1
SCHEMBL1760537 0.70 HMGCR (0.64) HMGCRESR1ESR2CNR1CNR2
SCHEMBL8013800 0.69 RXRA (0.51) HMGCRHSD17B1CYP1A2
SCHEMBL15867102 0.69 TYR (0.40) TRPA1CNR1CNR2TRPV1TRPV3
SCHEMBL1276072 0.68 CYP3A4 (0.49) HMGCRLMNAMAPTALDH1A1HTT
SCHEMBL11024762 0.68 HMGCR (0.61) HMGCRESR1ESR2CNR1CNR2
SCHEMBL11840310 0.66 HMGCR (0.59) HMGCRESR1ESR2CNR1CNR2
SCHEMBL4460505 0.66 HMGCR (0.42) HMGCRESR1ESR2ALOX5LMNA
SCHEMBL9722365 0.65 TP53 (0.33) ESR1ESR2TRPA1CNR1CNR2
SCHEMBL10459570 0.62 HMGCR (0.42) HMGCRLMNAMAPTALDH1A1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5149834-A Anticholesterol agent and enzyme inhibitors, for curing arteriosclerosis FUJIREBIO INC. (JP) 1992-09-22 US disclosed
EP-0445827-A2 4-Hydroxytetrahydropyran-2-one derivatives useful as cholesterol and lipid reducing agents FUJIREBIO INC. (JP) 1991-09-11 EP disclosed