SCHEMBL9723151

SCHEMBL9723151

CCc1ccc(C#N)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.37
TRPV4 Q9HBA0 1/20 0.35
CYP2A6 P11509 1/20 0.34
KCNJ1 P48048 1/20 0.34
AOC3 Q16853 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
EGLN2 Q96KS0 2/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
SLC22A12 Q96S37 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16428424 0.88 TRPV4 (0.35) TRPV4KCNJ1L3MBTL1TDP1EGLN2
SCHEMBL28574963 0.86 AR (0.36) ARTRPV4CYP2A6AOC3L3MBTL1
SCHEMBL16122697 0.84 AR (0.35) ARTRPV4CYP2A6KCNJ1AOC3
SCHEMBL9723274 0.84 AR (0.40) ARTRPV4KCNJ1L3MBTL1TDP1
SCHEMBL12763603 0.84 AR (0.38) ARTRPV4KCNJ1AOC3L3MBTL1
SCHEMBL23835170 0.82 GABRA1 (0.38) ARTRPV4CYP2A6AOC3L3MBTL1
SCHEMBL18552713 0.82 AR (0.44) ARKCNJ1AOC3
SCHEMBL12648422 0.82 GABRA1 (0.40) ARL3MBTL1TDP1
SCHEMBL6646922 0.81 TRPV4 (0.36) TRPV4L3MBTL1TDP1KDM4EHPGD
SCHEMBL14948935 0.80 AR (0.36) ARAOC3KDM4ECYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087764-A Deprotonation of a 1-substituted-2,3-difluorobenzene using an organometallic compound and reacting the reaction product with an electrophile Merck Patent Gesellschaft mit beschrankter Hafung (DE) 1992-02-11 US disclosed
EP-0363458-A1 2,3-DIFLUOROBENZENES. MERCK PATENT GMBH (DE) 1990-04-18 EP disclosed
CN-1037327-A Preparation 2, the method for 3-phenyl-difluoride class MERCK PATENT GMBH (DE) 1989-11-22 CN disclosed
WO-1989008629-A1 PROCESS FOR PREPARING 2,3-DIFLUOROBENZENES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-09-21 WO disclosed