SCHEMBL9724115

SCHEMBL9724115

C#CCN(Cc1ccc2ncc(N)c(Cl)c2c1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.66

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.66
TYMS P04818 5/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724117 0.92 DHFR (0.63) DHFRTYMS
SCHEMBL9724189 0.90 TYMS (0.72) DHFRTYMS
SCHEMBL9724232 0.86 DHFR (0.70) DHFRTYMS
SCHEMBL9724152 0.84 DHFR (0.67) DHFRTYMS
SCHEMBL9724262 0.84 DHFR (0.65) DHFRTYMS
SCHEMBL6579718 0.83 DHFR (0.78) DHFRTYMS
SCHEMBL9601470 0.83 TYMS (0.81) DHFRTYMS
SCHEMBL9724128 0.83 DHFR (0.70) DHFRTYMS
SCHEMBL9501327 0.82 DHFR (0.91) DHFRTYMS
SCHEMBL9224063 0.82 DHFR (0.91) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed