SCHEMBL9724152

SCHEMBL9724152

C#CCN(Cc1ccc2nc(Cl)cc(Cl)c2c1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.80

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.67
TYMS P04818 4/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724232 0.92 DHFR (0.70) DHFRTYMS
SCHEMBL9724311 0.91 DHFR (0.66) DHFRTYMS
SCHEMBL9729806 0.90 TYMS (0.63) DHFRTYMS
SCHEMBL9724197 0.90 DHFR (0.63) DHFRTYMS
SCHEMBL9724196 0.89 TYMS (0.73) TYMS
SCHEMBL9724117 0.87 DHFR (0.63) DHFRTYMS
SCHEMBL9724262 0.85 DHFR (0.65) DHFRTYMS
SCHEMBL6579718 0.85 DHFR (0.78) DHFRTYMS
SCHEMBL9724115 0.84 DHFR (0.66) DHFRTYMS
SCHEMBL9724128 0.84 DHFR (0.70) DHFRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed