SCHEMBL9724181

SCHEMBL9724181

NC(=O)Cc1cc(Cl)c2cc(CBr)ccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
NFKB1 P19838 1/20 0.35
STAT1 P42224 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
PLA2G10 O15496 2/20 0.34
CYP3A4 P08684 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724269 0.81 GRM2 (0.43) CYP4F2CYP4A11
SCHEMBL31434382 0.81 GRM2 (0.42) PLA2G10PLA2G2AKDM4E
SCHEMBL31434291 0.79 MEN1 (0.45) PLA2G10KDM4E
SCHEMBL9724221 0.79 KDM4E (0.40) CYP4F2CYP4A11HPGDCYP3A4CYP2C19
SCHEMBL9724211 0.79 NT5E (0.39) CYP4F2CYP4A11CYP3A4CYP2C19KDM4E
SCHEMBL9724264 0.78 CYP4F2 (0.41) CYP4F2CYP4A11NPC1RAB9ACYP3A4
SCHEMBL1599148 0.75 KDM4E (0.51) CYP4F2CYP4A11CYP3A4CYP2C19KDM4E
SCHEMBL9380126 0.72 LMNA (0.62) CYP4F2CYP4A11HPGDCYP3A4CYP2C19
SCHEMBL6604134 0.72 NPC1 (0.54) NPC1HPGDNFKB1STAT1RAB9A
SCHEMBL9383680 0.72 NPC1 (0.41) CYP4F2CYP4A11NPC1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed