SCHEMBL9724264

SCHEMBL9724264

CC(=O)OCc1cc(Cl)c2cc(CBr)ccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
ALDH1A1 P00352 2/20 0.38
CYP3A4 P08684 2/20 0.35
NOTUM Q6P988 1/20 0.34
PLA2G2A P14555 1/20 0.34
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34
CYP2C19 P33261 3/20 0.33
CYP1A2 P05177 2/20 0.33
CDK2 P24941 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HIF1A Q16665 1/20 0.33
NPC1 O15118 1/20 0.33
CYP2C9 P11712 1/20 0.33
RAB9A P51151 1/20 0.33
PKM P14618 1/20 0.33
ESRRB O95718 1/20 0.33
ESR1 P03372 1/20 0.33
ESRRA P11474 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724150 0.83 LMNA (0.51) ALDH1A1KDM4EPKMLMNA
SCHEMBL9724221 0.78 KDM4E (0.40) CYP4F2CYP4A11ALDH1A1CYP3A4CYP2C19
SCHEMBL9724181 0.78 PRKAB2 (0.36) CYP4F2CYP4A11CYP3A4PLA2G2ACYP2C19
SCHEMBL9724211 0.76 NT5E (0.39) CYP4F2CYP4A11CYP3A4CYP2C19KDM4E
SCHEMBL9555823 0.75 ALDH1A1 (0.44) ALDH1A1KDM4ENPC1RAB9ALMNA
SCHEMBL9383680 0.74 NPC1 (0.41) CYP4F2CYP4A11ALDH1A1KDM4ENPC1
SCHEMBL9382898 0.73 CYP4F2 (0.39) CYP4F2CYP4A11ALDH1A1CYP3A4KDM4E
SCHEMBL14358894 0.73 CYP1A2 (0.44) ALDH1A1CYP3A4PLA2G2ACYP2C19CYP1A2
SCHEMBL2671797 0.73 ELANE (0.41) ALDH1A1NOTUMCYP2C19CYP1A2NPC1
SCHEMBL336664 0.73 CYP4F2 (0.49) CYP4F2CYP4A11ALDH1A1CYP3A4NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed