SCHEMBL9724183

SCHEMBL9724183

Cc1cc(F)c2[nH]c(C)cc(=O)c2c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
HPGD P15428 6/20 0.44
KDM4E B2RXH2 5/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A2 P05177 2/20 0.42
GAA P10253 2/20 0.42
ADORA1 P30542 2/20 0.41
MAPT P10636 2/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
THRB P10828 1/20 0.37
ADORA2A P29274 1/20 0.37
GPR35 Q9HC97 1/20 0.35
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24533216 0.76 ALDH1A1 (0.58) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL22408257 0.72 KMT2A (0.33) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL17767227 0.71 F2 (0.37) ALDH1A1KDM4EMAPTLMNAHSD17B10
SCHEMBL21144481 0.71 HPGD (0.67) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL10005933 0.70 HPGD (0.70) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL22408085 0.68 GAA (0.33) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL22407860 0.68 ALDH1A1 (0.32) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL21886096 0.67 HRH4 (0.40) ALDH1A1KEAP1NFE2L2HPGDKDM4E
SCHEMBL16826531 0.67 KIF11 (0.50) ALDH1A1HPGDKDM4ESMN1; SMN2GAA
SCHEMBL28183336 0.66 ABCB1 (0.53) ALDH1A1HPGDKDM4ESMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed