SCHEMBL9724203

SCHEMBL9724203

Cc1cc(Cl)c2cc(C)c(C)cc2n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.63
LMNA P02545 1/20 0.60
POLB P06746 1/20 0.50
NR4A2 P43354 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
CYP1A2 P05177 3/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
RAD52 P43351 1/20 0.37
QRFPR Q96P65 1/20 0.37
NQO2 P16083 1/20 0.37
CRHR1 P34998 1/20 0.37
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 1/20 0.34
NCF1 P14598 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10519226 0.84 MAPT (0.56) MAPTLMNAPOLBNR4A2L3MBTL1
SCHEMBL5026883 0.84 MAPT (0.56) MAPTLMNAPOLBNR4A2L3MBTL1
SCHEMBL9724200 0.80 MAPT (0.51) MAPTLMNAPOLBNR4A2L3MBTL1
SCHEMBL5514349 0.80 MAPT (0.51) MAPTLMNAPOLBNR4A2L3MBTL1
SCHEMBL5522885 0.80 LMNA (0.53) MAPTLMNAPOLBNR4A2L3MBTL1
SCHEMBL10392506 0.79 CYP1A2 (0.56) MAPTLMNAPOLBNR4A2CYP1A2
SCHEMBL6605146 0.77 MAPT (0.49) MAPTLMNAPOLBALDH1A1SMN1; SMN2
SCHEMBL17372585 0.76 MAPT (0.56) MAPTLMNAPOLBALDH1A1KDM4E
SCHEMBL31353213 0.75 MAPT (0.50) MAPTLMNAPOLBNR4A2L3MBTL1
SCHEMBL4745343 0.75 POLB (0.72) MAPTLMNAPOLBNR4A2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed