SCHEMBL9724209

SCHEMBL9724209

CSc1cc(C)nc2ccc(C)cc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.59
CYP1A2 P05177 3/20 0.52
L3MBTL1 Q9Y468 2/20 0.51
KDM4E B2RXH2 4/20 0.45
ELANE P08246 1/20 0.43
HTT P42858 2/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ATM Q13315 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
PLK1 P53350 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MAPT P10636 2/20 0.41
JAK2 O60674 1/20 0.41
MITF O75030 1/20 0.41
KMT2A Q03164 1/20 0.41
PAX8 Q06710 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6848345 0.84 LMNA (0.53) LMNACYP1A2KDM4EHPGDHSD17B10
SCHEMBL6250314 0.81 KDM4E (0.64) LMNACYP1A2L3MBTL1KDM4EHPGD
SCHEMBL9724298 0.80 MAPT (0.40) LMNACYP1A2L3MBTL1KDM4EHPGD
SCHEMBL3531515 0.78 LMNA (0.66) LMNACYP1A2L3MBTL1KDM4EELANE
SCHEMBL6846717 0.77 KMT2A (0.52) LMNAL3MBTL1HTTHPGDMAPT
SCHEMBL30572382 0.74 LMNA (1.00) LMNACYP1A2L3MBTL1KDM4EELANE
SCHEMBL3760247 0.74 LMNA (0.61) LMNACYP1A2L3MBTL1KDM4EELANE
SCHEMBL29523105 0.74 LMNA (0.61) LMNACYP1A2L3MBTL1KDM4EELANE
SCHEMBL438604 0.74 NCF1 (0.63) LMNACYP1A2L3MBTL1KDM4EHSD17B10
SCHEMBL6766825 0.74 LMNA (0.61) LMNACYP1A2L3MBTL1KDM4EELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed