SCHEMBL9725906

SCHEMBL9725906

CCOC(=O)CNC1CCc2ccccc2C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.57
MTNR1B P49286 4/20 0.57
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
GRIN2B Q13224 4/20 0.50
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
THPO P40225 1/20 0.49
NPC1 O15118 1/20 0.49
MTOR P42345 1/20 0.49
RAB9A P51151 1/20 0.49
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
GMNN O75496 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9725905 0.99 MTNR1A (0.56) MTNR1AMTNR1BMAOAMAOBGRIN2B
SCHEMBL7334700 0.90 MTNR1A (0.47) MTNR1AMTNR1BGRIN2BKMT2APOLB
Hydrochloric Acid SCHEMBL7334726 0.89 MTNR1A (0.46) MTNR1AMTNR1BGRIN2BKMT2APOLB
Hydrochloric Acid SCHEMBL9545036 0.86 MTNR1A (0.56) MTNR1AMTNR1BMAOAMAOBGRIN2B
Hydrochloric Acid SCHEMBL9545040 0.86 MTNR1A (0.56) MTNR1AMTNR1BMAOAMAOBGRIN2B
SCHEMBL7926562 0.83 MTNR1A (0.64) MTNR1AMTNR1BCYP1A2CYP2C9
SCHEMBL11005303 0.83 DRD2 (0.58) MTNR1AMTNR1BGRIN2BKMT2APOLB
SCHEMBL11007069 0.83 DRD2 (0.65) MTNR1AMTNR1B
Hydrochloric Acid SCHEMBL11005295 0.82 DRD2 (0.57) MTNR1AMTNR1BGRIN2BKMT2APOLB
Hydrochloric Acid SCHEMBL11007066 0.82 DRD2 (0.63) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098892-A Angiotensin converting enzyme inhibitors as hypotensive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-03-24 US disclosed
US-4822818-A ANTIHYPERTENSIVE AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-04-18 US disclosed
US-4521607-A HYPOTENSIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1985-06-04 US disclosed
US-4474692-A L-Alanyl-N-(indan-2-yl)glycine, its esters and salts thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1984-10-02 US disclosed
EP-0051391-B1 BICYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1984-09-05 EP disclosed
EP-0051391-A1 Bicyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1982-05-12 EP disclosed
EP-0035868-A1 Bicyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1981-09-16 EP disclosed