SCHEMBL9725938

SCHEMBL9725938

CCOC(=O)CCNC1Cc2ccccc2C1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.48
MTNR1A P48039 2/20 0.48
MTNR1B P49286 2/20 0.48
GRIN2B Q13224 3/20 0.46
TOP2A P11388 1/20 0.46
NOTUM Q6P988 1/20 0.45
SIGMAR1 Q99720 1/20 0.44
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.42
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9725932 0.99 NAMPT (0.47) NAMPTMTNR1AMTNR1BGRIN2BTOP2A
SCHEMBL24651033 0.92 NAMPT (0.52) NAMPTMTNR1AMTNR1BGRIN2BTOP2A
SCHEMBL24651034 0.86 GRIN2B (0.50) MTNR1AMTNR1BGRIN2BNOTUMSIGMAR1
SCHEMBL7334700 0.85 MTNR1A (0.47) NAMPTMTNR1AMTNR1BGRIN2BALDH1A1
Hydrochloric Acid SCHEMBL7334726 0.84 MTNR1A (0.46) NAMPTMTNR1AMTNR1BGRIN2BALDH1A1
SCHEMBL18983637 0.79 DRD3 (0.60) GRIN2B
SCHEMBL24651031 0.78 GRIN2B (0.59) MTNR1AMTNR1BGRIN2BSIGMAR1ALDH1A1
SCHEMBL8309501 0.78 GRIN2B (0.53) MTNR1AMTNR1BGRIN2BNOTUMSIGMAR1
SCHEMBL7140606 0.77 SMYD3 (0.50) TOP2AALDH1A1GAAKDM4ELMNA
SCHEMBL10531104 0.77 NOTUM (0.48) NAMPTNOTUMCYP4F2CYP4A11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022238507-A1 THERAPEUTIC AMINOINDANE COMPOUNDS AND COMPOSITIONS AWAKN LS EUROPE HOLDINGS LIMITED (IE) 2022-11-17 WO disclosed
US-5098892-A Angiotensin converting enzyme inhibitors as hypotensive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-03-24 US disclosed
US-4822818-A ANTIHYPERTENSIVE AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-04-18 US disclosed
US-4474692-A L-Alanyl-N-(indan-2-yl)glycine, its esters and salts thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1984-10-02 US disclosed
EP-0051391-B1 BICYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1984-09-05 EP disclosed
EP-0051391-A1 Bicyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1982-05-12 EP disclosed