SCHEMBL9726439

SCHEMBL9726439

CCCN(CCC)Cc1ccc(CNC)cc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.64
LOXL2 Q9Y4K0 1/20 0.48
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.43
CYP3A4 P08684 1/20 0.43
RORC P51449 2/20 0.42
BCHE P06276 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1206283 0.80 HRH3 (0.64) HRH3MAPTRORCBCHE
SCHEMBL20287494 0.77 HRH3 (0.72) HRH3MAPTRORCBCHECYP1A2
Water SCHEMBL28117059 0.77 HRH3 (0.65) HRH3MAPTKDM4ERORCBCHE
SCHEMBL19088665 0.76 HRH3 (0.64) HRH3LOXL2MAPTRORCBCHE
SCHEMBL11529383 0.76 LOXL2 (0.44) LOXL2MAPTKDM4ECYP3A4NPSR1
SCHEMBL11402252 0.76 HRH3 (0.53) HRH3RORCBCHE
SCHEMBL14640185 0.75 HRH3 (0.69) HRH3MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL996084 0.75 HRH3 (0.63) HRH3MAPTBCHECYP1A2CYP2D6
SCHEMBL1204908 0.75 HRH3 (0.69) HRH3MAPTCYP3A4RORCBCHE
SCHEMBL13078725 0.75 HRH3 (0.69) HRH3MAPTBCHECYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed