SCHEMBL9726454

SCHEMBL9726454

[CH]=CC(=O)NCCC(=O)OCC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.45
MGAM O43451 1/20 0.45
SI P14410 1/20 0.45
MGAM2 Q2M2H8 1/20 0.45
ALDH1A1 P00352 4/20 0.42
TRPA1 O75762 1/20 0.42
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 2/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
NR1I2 O75469 1/20 0.38
PGR P06401 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
PTGS2 P35354 1/20 0.38
PDE4D Q08499 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TOP2A P11388 1/20 0.37
MLYCD O95822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726435 0.82 TSHR (0.48) ALDH1A1KMT2AMAPTHPGDTSHR
SCHEMBL26478848 0.81 ZDHHC20 (0.50) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL9726440 0.81 GAA (0.52) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL7088568 0.78 GAA (0.54) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL15201482 0.76 GAA (0.52) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL1425763 0.76 GAA (0.52) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL48439 0.76 GAA (0.52) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL8634353 0.76 ZDHHC20 (0.45) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL4093617 0.76 CYP1A2 (0.47) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL3553857 0.76 TRPA1 (0.54) GAAMGAMSIMGAM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed