SCHEMBL9726460

SCHEMBL9726460

O=C(c1ccc(C(F)(F)F)cc1)c1ccc(Cl)cc1Cl

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.64
MAPT P10636 1/20 0.59
RAB9A P51151 1/20 0.59
CYP2C8 P10632 1/20 0.50
CCR9 P51686 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
TSHR P16473 1/20 0.49
CASP1 P29466 1/20 0.49
HTT P42858 1/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
GRIK1 P39086 1/20 0.47
P2RX1 P51575 1/20 0.47
P2RX4 Q99571 1/20 0.47
P2RX7 Q99572 1/20 0.47
TMPRSS4 Q9NRS4 1/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
CYP2C9 P11712 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8005994 0.86 CYP2C8 (0.49) SRD5A2MAPTRAB9ACYP2C8CCR9
SCHEMBL25042900 0.84 CYP2C8 (0.48) SRD5A2MAPTRAB9ACYP2C8CCR9
SCHEMBL9496067 0.84 SRD5A2 (0.79) SRD5A2MAPTRAB9ASMN1; SMN2TSHR
SCHEMBL15391539 0.82 CES2 (0.50) SRD5A2MAPTRAB9ASMN1; SMN2TSHR
SCHEMBL611648 0.81 SRD5A2 (0.70) SRD5A2MAPTRAB9ASMN1; SMN2TSHR
SCHEMBL10396396 0.81 RECQL (0.53) SRD5A2MAPTCYP2C8CCR9TSHR
SCHEMBL7995549 0.81 CYP2C8 (0.45) SRD5A2MAPTRAB9ACYP2C8CCR9
SCHEMBL11057221 0.81 SRD5A2 (0.68) SRD5A2CES2CES1ESR1MAPK1
SCHEMBL8437570 0.80 SRD5A2 (0.96) SRD5A2MAPTRAB9ASMN1; SMN2TSHR
SCHEMBL610783 0.80 SRD5A2 (0.72) SRD5A2MAPTRAB9ASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed