SCHEMBL9726515

SCHEMBL9726515

Cc1cc(F)ccc1C(=Cc1nnnn1C)c1ccc(F)cc1C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.39
ALDH1A1 P00352 3/20 0.34
SLC6A1 P30531 3/20 0.33
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PKM P14618 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726825 0.86 ALDH1A1 (0.39) ALDH1A1NPC1LMNARAB9ASMN1; SMN2
SCHEMBL8846423 0.81 ALDH1A1 (0.41) ESR1ALDH1A1LMNARAB9ASMN1; SMN2
SCHEMBL9726750 0.81 ALDH1A1 (0.33) ESR1ALDH1A1NPC1LMNARAB9A
SCHEMBL9726395 0.78 SRC (0.34) ESR1ALDH1A1SMN1; SMN2
SCHEMBL9726766 0.76 PTGS2 (0.44) ALDH1A1RAB9ASMN1; SMN2PKM
SCHEMBL9726776 0.76 PTGS2 (0.44) ALDH1A1RAB9ASMN1; SMN2PKM
SCHEMBL9726773 0.76 PTGS2 (0.44) ALDH1A1RAB9ASMN1; SMN2PKM
SCHEMBL10610927 0.74 ESR1 (0.44) ESR1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL10610936 0.74 ESR1 (0.44) ESR1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL9726576 0.71 HMGCR (0.41) ESR1ALDH1A1NPSR1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US claimed
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4939265-A Intermediates and process for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-07-03 US disclosed
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed