SCHEMBL9726523

SCHEMBL9726523

COc1ccc(C(=O)c2ccccc2C(F)(F)F)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.56
LMNA P02545 3/20 0.53
MAPT P10636 2/20 0.53
GAA P10253 2/20 0.53
ATM Q13315 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C19 P33261 2/20 0.51
HPGD P15428 2/20 0.51
PGR P06401 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
AR P10275 1/20 0.51
CHRM1 P11229 1/20 0.51
ALOX15 P16050 1/20 0.51
TBXA2R P21731 1/20 0.51
SLC6A2 P23975 1/20 0.51
ADRA1A P35348 1/20 0.51
HIF1A Q16665 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1407535 0.88 NPC1 (0.52) NPC1LMNAMAPTGAAATM
SCHEMBL8760033 0.86 LMNA (0.71) NPC1LMNAMAPTGAAATM
SCHEMBL28899309 0.85 NPC1 (0.58) NPC1LMNAMAPTGAAATM
SCHEMBL3236831 0.84 NPC1 (0.68) NPC1LMNAMAPTGAASMN1; SMN2
SCHEMBL7181308 0.84 NPC1 (0.45) NPC1LMNAMAPTGAAATM
SCHEMBL285924 0.82 NPC1 (0.79) NPC1LMNAMAPTGAASMN1; SMN2
SCHEMBL31575666 0.82 NPC1 (0.79) NPC1LMNAMAPTGAASMN1; SMN2
SCHEMBL4935615 0.81 NPC1 (0.60) NPC1LMNAMAPTGAASMN1; SMN2
SCHEMBL7479627 0.80 KMT2A (0.60) NPC1LMNAMAPTSMN1; SMN2NPSR1
SCHEMBL15125786 0.80 NPC1 (0.62) NPC1LMNAMAPTGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed