SCHEMBL9726581

SCHEMBL9726581

CCOc1cccc(CNc2cnn(CC)c(=O)c2Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.54
BRD9 Q9H8M2 3/20 0.54
BPTF Q12830 2/20 0.53
KAT2B Q92831 3/20 0.50
MAPT P10636 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.41
NPBWR1 P48145 1/20 0.41
P2RX7 Q99572 1/20 0.40
GRM2 Q14416 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE9A O76083 1/20 0.39
CYP3A4 P08684 2/20 0.39
NR3C1 P04150 1/20 0.39
ROCK2 O75116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726627 0.92 BRD4 (0.52) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL9726399 0.88 BRD4 (0.49) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL9726483 0.87 BRD4 (0.41) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL9726528 0.85 BRD4 (0.52) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL10601520 0.84 BRD4 (0.74) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL9726487 0.83 BRD4 (0.50) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL9726575 0.80 BRD4 (0.47) BRD4BRD9BPTFKAT2BGRM2
SCHEMBL9726489 0.79 ALDH1A1 (0.46) BRD4BRD9BPTFKAT2BMAPT
SCHEMBL9726443 0.79 BACE1 (0.43) BRD4BRD9BPTFALDH1A1GRM2
SCHEMBL9726619 0.76 BRD4 (0.49) BRD4BRD9BPTFKAT2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US claimed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP claimed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP claimed