SCHEMBL9726718

SCHEMBL9726718

COc1ccc(C(=C(/C=C/C=O)c2nnnn2C)c2ccc(OC)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.43
ALDH1A1 P00352 5/20 0.42
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPT P10636 1/20 0.36
HIF1A Q16665 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TCF4 P15884 1/20 0.36
CTNNB1 P35222 1/20 0.36
ERCC5 P28715 1/20 0.36
FEN1 P39748 1/20 0.36
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726725 1.00 HMGCR (0.43) HMGCRALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL9726963 0.87 TCF4 (0.46) HMGCRALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL9726481 0.85 HMGCR (0.57) HMGCRALDH1A1
SCHEMBL9726476 0.85 HMGCR (0.57) HMGCRALDH1A1
SCHEMBL9726855 0.85 HMGCR (0.43) HMGCRALDH1A1RAB9ASMN1; SMN2POLB
SCHEMBL9726851 0.85 HMGCR (0.43) HMGCRALDH1A1RAB9ASMN1; SMN2POLB
SCHEMBL9727124 0.81 HMGCR (0.53) HMGCRALDH1A1
SCHEMBL9726717 0.81 HMGCR (0.53) HMGCRALDH1A1
SCHEMBL9799413 0.81 HMGCR (0.55) HMGCRALDH1A1
SCHEMBL9799408 0.81 HMGCR (0.55) HMGCRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US claimed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO claimed
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed