SCHEMBL9726855

SCHEMBL9726855

Cn1nnnc1C(C=CC=O)=C(c1ccccc1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.43
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RECQL P46063 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726851 1.00 HMGCR (0.43) HMGCRNPC1RAB9ANFKB1NFKB2
SCHEMBL9727128 0.93 HMGCR (0.53) HMGCRALDH1A1
SCHEMBL9726717 0.93 HMGCR (0.53) HMGCRALDH1A1
SCHEMBL9727124 0.93 HMGCR (0.53) HMGCRALDH1A1
SCHEMBL9726481 0.87 HMGCR (0.57) HMGCRALDH1A1
SCHEMBL9726476 0.87 HMGCR (0.57) HMGCRALDH1A1
SCHEMBL9726944 0.86 HMGCR (0.42) HMGCRRAB9AALDH1A1RECQLPOLB
SCHEMBL9726718 0.85 HMGCR (0.43) HMGCRRAB9AALDH1A1SMN1; SMN2POLB
SCHEMBL9726725 0.85 HMGCR (0.43) HMGCRRAB9AALDH1A1SMN1; SMN2POLB
SCHEMBL9799413 0.82 HMGCR (0.55) HMGCRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US claimed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO claimed
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4898949-A Intermediates for the preparation of antihypercholesterolemic tetrazole compounds BRISTOL-MYERS COMPANY (US) 1990-02-06 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed