SCHEMBL9727111

SCHEMBL9727111

C[CH]SC(=O)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.48
CES1 P23141 3/20 0.48
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
MAPT P10636 4/20 0.43
HPGD P15428 2/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX12 P18054 1/20 0.43
CYP2C19 P33261 1/20 0.43
GSK3B P49841 2/20 0.42
SRD5A2 P31213 1/20 0.42
MAPK1 P28482 1/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727180 0.76 CES2 (0.54) CES2CES1ALOX15TSHRCA1
SCHEMBL8716211 0.75 CES2 (0.59) CES2CES1ALOX15TSHRCA1
SCHEMBL13571696 0.75 CES2 (0.59) CES2CES1ALOX15TSHRCA1
SCHEMBL2915596 0.71 CYP1A2 (0.57) CES2CES1ALOX15TSHRCA1
SCHEMBL9727178 0.71 CES2 (0.54) CES2CES1ALOX15TSHRCA1
SCHEMBL9727115 0.71 HDAC3 (0.57) CES2CES1ALOX15TSHRCA1
SCHEMBL27870723 0.70 CES2 (0.52) CES2CES1ALOX15TSHRCA1
SCHEMBL28629808 0.68 MAPT (0.63) CES2CES1MAPTHPGDCYP1A2
SCHEMBL13960902 0.68 MAPT (0.63) CES2CES1MAPTHPGDCYP1A2
SCHEMBL11424462 0.68 GSK3B (0.54) CES2CES1ALOX15TSHRCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5144027-A Cephalosporins, process for producing the same, intermediates thereof and process for producing the intermediates TOYAMA CHEMICAL CO., LTD. (JP) 1992-09-01 US disclosed
US-4879381-A ANTIBIOTICS TOYOMA CHEMICAL COMPANY, LTD. (JP) 1989-11-07 US disclosed
US-4717767-A ANTIBIOTICS TOYAMA CHEMICAL CO., LTD. (JP) 1988-01-05 US disclosed
US-4698352-A 4-oxo-1,4-dihydronicotinic acid derivatives, salts thereof, and antibacterial agents containing the same TOYAMA CHEMICAL CO., LTD. (JP) 1987-10-06 US disclosed
US-4673738-A Novel intermediates of cephalosporins and process for producing 7-(substituted or unsubstituted amino)-3-substituted methyl-Δ3 -cephem-4-carboxylic acids HANDI-PAC INC. (US) 1987-06-16 US disclosed
US-4618606-A Antibiotic 7-(thiazolyl)-3-(pyrazinylmethyl) or (pyridazinylmethyl) cephalosporins TOYAMA CHEMICAL CO., LTD. (JP) 1986-10-21 US disclosed
US-4489072-A BACTERICIDE, ANTIBIOTIC TOYAMA CHEMICAL CO., LTD. (JP) 1984-12-18 US disclosed